Lappaconitine hydrobromide is a C19-diterpenoid alkaloid hydrobromide salt. It acts as a voltage-gated sodium channel (Nav1.5, Nav1.7) blocker.

Scopolamine butylbromide is an active cholinergic receptor antagonist that binds with high affinity to M2 and M3 muscarinic receptors.

Vinblastine sulfate is a cytotoxic alkaloid that inhibits the formation of microtubule and suppresses nAChR.

Thapsigargin, an endoplasmic reticulum (ER) stress inducer, is a microsomal Ca2+-ATPase inhibitor.

Vinorelbine ditartrate is an anti-mitotic agent which inhibits the proliferation of Hela cells.

Eupatilin, a lipophilic flavonoid, is a PPARα agonist.

Cytisine is an alkaloid and a partial agonist of α4β2 nAChRs, with partial to full agonism at β4-containing receptors and α7 receptors.

Digoxin is a potent inhibitor of Na+/K+-ATPase.

Scopolamine hydrobromide is a high-affinity muscarinic antagonist that can cross the blood-brain barrier.

Xanthotoxin is a furanocoumarin compound and a cytochrome P450 inhibitor.

Lovastatin is a cell-permeable HMG-CoA reductase inhibitor.

Eriodictyol is an active TRPV1 receptor antagonist.

Ursodeoxycholic acid is a secondary bile acid issued from the transformation of (cheno)deoxycholic acid by intestinal bacteria, acting through interactions with bile acid-activated receptors including TGR5 and FXR.

Triptolide is a diterpenoid triepoxide and acts as an NF-κB activation inhibitor.

1-Chloroethyl palmitate is a long-chain fatty acid ester featuring a C16 hydrophobic fatty chain and a chloroethyl reactive site; it can be used in the development of lipid derivatives and functionalized ester intermediates.

Podofilox (Podophyllotoxin) is a potent inhibitor of microtubule assembly and DNA topoisomerase II.