Anisatin, a pure toxic substance isolated from the seeds of Illicium anisatum acts as a picrotoxin-like, non-competitive GABA antagonist.

Potassium Hydroxycitrate is an multi-target, multi-bioactive organic acid.

Isosakuranetin is a flavanone flavonoid which can be found in the fruit of Citrus bergamia. Isosakuranetin is a TRPM3 blocker.

Anisodamine is a belladonna alkaloid, is a non-subtype-selective muscarinic, and also a nicotinic cholinoceptor antagonist.

Kaempferitrin is a natural flavonoid, possesses antinociceptive.

Cholest-4,6-diene-3-ol belongs to the class of sterol derivatives associated with cholesterol oxidation or dehydrogenation.

Cornuside is an iridoid glycoside,and it is also an inhibitor.

Nevadensin is a natural flavonoid, is a selective human carboxylesterase 1 (hCE1) inhibitor, Nevadensin has a variety of pharmacological effects.

Sappanone A is an homoisoflavone found in sappan L. Sappanone A is a PDE4 and NF-κB inhibitor.

Stachydrine is a major constituent of Chinese herb leonurus heterophyllus sweet used to promote blood circulation and dispel blood stasis.

Gartanin is a natural xanthone of mangosteen, Gartanin is also an inhibitor.

Adenanthin is a natural flavonoid product.

Sempervirine Nitrate is an alkaloid derived from Gelsemium elegans Benth.

Valerenic Acid, a sesquiterpenoid, is an positive allosteric modulator of GABAA receptors.

Cucurbitacin S is isolated from the Cucurbitaceae family.

Chelerythrine Chloride is a potent, cell-permeable inhibitor of protein kinase C.