需要帮助?我们经验深厚的专家团队,随时为您提供全力支持。
产品编号
AKA-384
CAS号码
856867-55-5
分子式
C17H16FN6O6P
分子量
Tedizolid phosphate
磷酸泰地唑胺
Tedizolid phosphate
856867-55-5
C17H16FN6O6P
450.32
98.0%~102.0%
磷酸泰地唑胺是一种噁唑烷酮环、含氟芳基及四唑杂环结构的抗菌药物前药,是 MAO-A 和 MAO-B 抑制剂。 包装: 1kg/袋,5kg/袋,25kg/袋 供货情况: 现货供应 API Current Development Status: A3---Process Development / Scale-Up Reference: Aktin major API development processes: A1.Feasibility / Route Development A2.Laboratory Process Development A3.Process Development / Scale-Up A4.GMP Clinical Development A5.Commercial GMP Supply
[1].Im WB, Choi SH, Park JY, Choi SH, Finn J, Yoon SH. Discovery of torezolid as a novel 5-hydroxymethyl-oxazolidinone antibacterial agent. Eur J Med Chem. 2011;46(4):1027-1039. doi:10.1016/j.ejmech.2011.01.014
[2].Lei Y, Jin B, Ma C, Zhang T, Li T. Identification of forced degradation products of tedizolid phosphate by liquid chromatography/electrospray ionization tandem mass spectrometry. J Pharm Biomed Anal. 2017;139:221-231. doi:10.1016/j.jpba.2017.03.006
[3].Prokocimer P, Bien P, DeAnda C, Pillar CM, Bartizal K. In vitro activity and microbiological efficacy of tedizolid (TR-700) against Gram-positive clinical isolates from a phase 2 study of oral tedizolid phosphate (TR-701) in patients with complicated skin and skin structure infections. Antimicrob Agents Chemother. 2012;56(9):4608-4613. doi:10.1128/AAC.00458-12
关于仿制药原料药(generic APIs)的信息仅供一般参考和市场评估之用。监管状态、市场适用性、质量标准、专利及商业条款可能因国家/地区而异,并可能随时间变化。用户在作出任何监管、生产、投资或商业决策之前,应自行向相关监管机构及专业人士核实所有信息。 我们不向个人提供产品或服务。请严格遵守所有适用法律、法规,并仅按承诺用途使用相关产品或服务;严禁用于任何其他目的。
*本产品不用于诊断、治疗、治愈或预防任何疾病,仅供科研研究使用。