Lovastatin
Cat. No.
AKA-69
CAS No.
75330-75-5
MF
C24H36O5
MW
404.5396
Lovastatin is a cell-permeable HMG-CoA reductase inhibitor.
Xanthotoxin
Cat. No.
AKA-70
CAS No.
298-81-7
MF
C12H8O4
MW
216.1895
Xanthotoxin is a furanocoumarin compound and a cytochrome P450 inhibitor.
Scopolamine Hydrobromide
Cat. No.
AKA-80
CAS No.
114-49-8
MF
C17H22BrNO4
MW
384.26488
Scopolamine hydrobromide is a high-affinity muscarinic antagonist that can cross the blood-brain barrier.
Digoxin
Cat. No.
AKA-81
CAS No.
20830-75-5
MF
C41H64O14
MW
780.93846
Digoxin is a potent inhibitor of Na+/K+-ATPase.
Cytisine
Cat. No.
AKA-91
CAS No.
485-35-8
MF
C11H14N2O
MW
190.24
Cytisine is an alkaloid and a partial agonist of α4β2 nAChRs, with partial to full agonism at β4-containing receptors and α7 receptors.
Eupatilin
Cat. No.
AKA-94
CAS No.
22368-21-4
MF
C18H16O7
MW
344.31
Eupatilin, a lipophilic flavonoid, is a PPARα agonist.
Vinorelbine Tartrate
Cat. No.
AKA-95
CAS No.
125317-39-7
MF
C53H66N4O20
MW
1079.1
Vinorelbine ditartrate is an anti-mitotic agent which inhibits the proliferation of Hela cells.
Thapsigargin
Cat. No.
AKA-97
CAS No.
67526-95-8
MF
C34H50O12
MW
650.8
Thapsigargin, an endoplasmic reticulum (ER) stress inducer, is a microsomal Ca2+-ATPase inhibitor.
Vinblastine Sulfate
Cat. No.
AKA-102
CAS No.
143-67-9
MF
C46H58N4O9.H2O4S
MW
909.1
Vinblastine sulfate is a cytotoxic alkaloid that inhibits the formation of microtubule and suppresses nAChR.
Scopolamine Butylbromide
Cat. No.
AKA-103
CAS No.
149-64-4
MF
C21H30BrNO4
MW
440.4
Scopolamine butylbromide is an active cholinergic receptor antagonist that binds with high affinity to M2 and M3 muscarinic receptors.
Lappaconitine Hydrobromide
Cat. No.
AKA-104
CAS No.
97792-45-5
MF
C32H45BrN2O8
MW
665.6
Lappaconitine hydrobromide is a C19-diterpenoid alkaloid hydrobromide salt. It acts as a voltage-gated sodium channel (Nav1.5, Nav1.7) blocker.
Vincristine Sulfate
Cat. No.
AKA-105
CAS No.
2068-78-2
MF
C46H58N4O14S
MW
923
Vincristine sulfate is a microtubule inhibitor that binds β-tubulin and disrupts microtubule polymerization.
Boldine
Cat. No.
AKA-108
CAS No.
476-70-0
MF
C19H21NO4
MW
327.37
Boldine is an apomorphine isoquinoline alkaloid.
Scopolamine Hydrochloride
Cat. No.
AKA-118
CAS No.
55-16-3
MF
C17H22ClNO4
MW
339.8
Scopolamine hydrochloride is a high-affinity muscarinic antagonist that can cross the blood-brain barrier.
Resiniferatoxin
Cat. No.
AKA-119
CAS No.
57444-62-9
MF
C37H40O9
MW
628.71
Resiniferatoxin is a selective agonist of the transient receptor potential vanilloid 1 (TRPV1) receptor.
Hypericin Sodium
Cat. No.
AKA-120
CAS No.
144788-48-7
MF
C30H16O8.Na
MW
527.43
Hypericin Sodium exhibits good water dispersibility and solubility in organic solvents. It is a potent photosensitizer. Hypericin sodium also acts as an inhibitor of various enzymes including monoamine oxidase (MAO), protein kinase C (PKC), and reverse transcriptase.